RS-93522 - CAS 104060-12-0

RS-93522 is an antagonist of calcium channel. RS-93522 had the additional property of inhibiting phosphodiesterase activity in myocardial homogenates (IC50 = 1.6 x 10 (-5) M), the potency and efficacy of phosphodiesterase inhibition was similar to that for milrinone in the same system. As expected of Ca channel antagonists, it has a negative inotropic effect on cultured myocardial cells.

Others, Calcium Channel

Membrane transporter/Ion channel, Others, Metabolism

104048

C27H30N2O9

526.54

C(OCCC1=CC=C(OCC(CO)O)C=C1)(=O)C=2C(C(C(OC)=O)=C(C)NC2C)C3=CC(N(=O)=O)=CC=C3

-20°C

Ice Packs

Small Compound