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Rucaparib camsylate - CAS 1327258-57-0
Rucaparib camsylate - CAS 1327258-57-0
SKU:MF-0049452-01
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Product Details
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Bioactivity
Rucaparib (AG014699) camsylate is an orally active inhibitor of PARP proteins (PARP-1, PARP-2, and PARP-3) with a Ki=1.4 nM for PARP-1, and also inhibits hexose hexaphosphate dehydrogenase (H6PD) . Rucaparib camsylate has potential for investigation in debulking resistant prostate cancer (CRPC) studies.
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Target
PARP, Others
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Related Pathways
DNA Damage/DNA Repair, Others, Chromatin/Epigenetic
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CAS Number
1327201
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Molecular Formula
C19H18FN3O.xC10H16O4S
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Storage Temperature
-20°C
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Shipping Conditions
Ice Packs
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Category
Small Compound