SR-12062 - CAS 1623019-77-1

SR-12062 functions as a full agonist at neurotensin receptor 1 (NTSR1), demonstrating notable efficacy and increased potency. Its EC50 value on NTSR1 is 2 μM, with complete receptor activation (Emax=100%) . Compared to the parent compound 1 (EC50=178 μM; Emax=17%), SR-12062 shows approximately 90-fold greater potency.

1622941

C25H25N3O3

415.48

C(C(N[C@@H](CC(C)C)C(O)=O)=O)N1C=2C(=CC(=CC2)C3=CC4=C(N=C3)C=CC=C4)C=C1

-20°C

Ice Packs

Small Compound