SRA880 free base - CAS 187218-90-2

SRA880 is a non-peptide antagonist of somatostatin sst1-receptor. SRA880 displayed significantly lower affinity for the other human recombinant somatostatin receptors (pK (d) < or = 6.0) . SRA880 shows a certain binding affinity to the human dopamine D4 receptors. SRA880 positively modulates release of endogenous SRIF, was found to synergize with imipramine in causing antidepressant-like effects in the tail suspension test.

Others, Somatostatin

Others, GPCR/G Protein

187126

C26H32N4O4

464.56

O=[N+](C(C=C1)=CC=C1N(CC2)CCN2C([C@@H](C3)C[C@@](CC4=C(OC)C=CC=C4C5)([H])[C@]5([H])N3C)=O)[O-]

-20°C

Ice Packs

Small Compound