SSR240612 - CAS 464930-42-5

SSR240612 is a potent, orally active, specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 nM for B1 receptors and 358-481 nM for B2 receptors, respectively) .

Bradykinin Receptor

GPCR/G Protein

464930-42-5

0.9916

C42H53ClN4O7S

793.41

Cl.COc1ccc2cc(ccc2c1)S(=O)(=O)N[C@H](CC(=O)N[C@H](Cc1ccc(CN2[C@@H](C)CCC[C@H]2C)cc1)C(=O)N(C)C(C)C)c1ccc2OCOc2c1

-20°C

Ice Packs

Small Compound