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Molfinity

TAK-243 - CAS 1450833-55-2

TAK-243 - CAS 1450833-55-2

MF-0034114-01

$40.65 USD
$40.65 USD
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Product Details

  • Bioactivity

    TAK-243 (MLN7243) is a selective inhibitor of the ubiquitin-activating enzyme UAE (IC50=1 nM), blocking ubiquitin binding and disrupting both mono-ubiquitin signaling and overall protein ubiquitination. TAK-243 exhibits antitumor activity and promotes apoptosis.

  • Target

    NF-κB, Apoptosis, E1/E2/E3 Enzyme

  • Related Pathways

    Apoptosis, NF-κB, Ubiquitination

  • CAS Number

    1450776

  • Purity

    0.9893

  • Molecular Formula

    C19H20F3N5O5S2

  • Molecular Weight

    519.52

  • SMILES

    NS(=O)(=O)OC[C@H]1C[C@@H](Nc2ccnc3cc(nn23)-c2cccc(SC(F)(F)F)c2)[C@H](O)[C@@H]1O

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound