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Tazemetostat hydrobromide - CAS 1467052-75-0

Tazemetostat hydrobromide - CAS 1467052-75-0

MF-0019340-01

$36.91 USD
$36.91 USD
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Product Details

  • Bioactivity

    Tazemetostat hydrobromide (E-7438 hydrobromide) is a potent and selective EZH2 inhibitor. Tazemetostat hydrobromide inhibits the activity of human polycomb repressive complex 2 (PRC2) -containing wild-type EZH2 (Ki: 2.5 nM) . Tazemetostat hydrobromide also inhibits EZH1 (IC50: 392 nM) .

  • Target

    Histone Methyltransferase

  • Related Pathways

    Chromatin/Epigenetic

  • CAS Number

    1466977

  • Purity

    0.998

  • Molecular Formula

    C34H45BrN4O4

  • Molecular Weight

    653.65

  • SMILES

    O=C(C1=CC(C2=CC=C(CN3CCOCC3)C=C2)=CC(N(CC)C4CCOCC4)=C1C)NCC5=C(C)C=C(C)NC5=O.[H]Br

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound