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Tazemetostat trihydrochloride - CAS 1403255-00-4

Tazemetostat trihydrochloride - CAS 1403255-00-4

MF-0032816-01

$1,480.33 USD
$1,480.33 USD
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Product Details

  • Bioactivity

    Tazemetostat trihydrochloride is a selective and orally available inhibitor of EZH2 (IC50: 4 nM for rat EZH2) . It inhibits the activity of human PRC2-containing wild-type EZH2 (Ki: 2.5 nM) . It inhibits EZH2 (IC50s: 11 and 16 nM in peptide assay and nucleosome assay) .

  • Target

    Histone Methyltransferase

  • Related Pathways

    Chromatin/Epigenetic

  • CAS Number

    1403255-00-4

  • Molecular Formula

    C34H47Cl3N4O4

  • Molecular Weight

    682.12

  • SMILES

    O=C(C1=CC(C2=CC=C(CN3CCOCC3)C=C2)=CC(N(C4CCOCC4)CC)=C1C)NCC5=C(C)C=C(C)NC5=O.Cl.Cl.Cl

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound