TGR5 Receptor Agonist 4 - CAS 1872436-42-4

TGR5 Receptor Agonist 4, a selective agonist for the Bile Acid Receptor (TGR5), exhibits potent activity with an EC50 of 2 nM for human TGR5 (hTGR5) and 3 nM for mouse TGR5 (mTGR5) . It is notably involved in mediating hypoglycemic and weight loss effects [1].

Others, GPCR19

GPCR/G Protein, Others

1872436-42-4

C25H27ClN2O5

470.95

C(OCC1=C(OC)C=CC=C1)(=O)C=2[C@@H](CC(=O)N(C[C@H]3CCCO3)C2C)C=4C=CC(Cl)=NC4

-20°C

Ice Packs

Small Compound