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Molfinity

TP-064 - CAS 2080306-20-1

TP-064 - CAS 2080306-20-1

SKU:MF-0013770-01

Regular price $33.92 USD
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  • Bioactivity

    TP-064 is a potent and selective PRMT4 inhibitor, featuring an IC50 < 10nM for methylation of H3 (1-25) and over 100-fold selectivity compared to other histone methyltransferases and non-epigenetic targets. It inhibits the methylation of MED12 in cells with an IC50 of 43 nM.

  • Target

    Histone Methyltransferase

  • Related Pathways

    Chromatin/Epigenetic

  • CAS Number

    2080285

  • Purity

    0.9907

  • Molecular Formula

    C28H34N4O2

  • Molecular Weight

    458.6

  • SMILES

    CNCCN1CCC(CC1)c1cc(CN(C)C(=O)c2cccc(Oc3ccccc3)c2)ccn1

  • Storage Temperature

    -20°C

  • Shipping Conditions

    Ice Packs

  • Category

    Small Compound