TRV-120027 acetate (1234510-46-3 free base) - CAS 1824712-70-0

TRV-120027 acetate is a β-arrestin-1-biased agonist of the angiotensin II receptor type 1 (AT1 receptor) and engages -arrestins while blocking G-protein signaling.

RAAS, Arrestin

Endocrinology/Hormones, GPCR/G Protein

1824642

0.9934

C45H71N13O12

986.14

CC(O)=O.C[C@H](C(O)=O)NC([C@H]1N(C([C@H](CC2=CNC=N2)NC([C@H]([C@@H](C)CC)NC([C@H](CC3=CC=C(O)C=C3)NC([C@H](C(C)C)NC([C@H](CCCNC(N)=N)NC(CNC)=O)=O)=O)=O)=O)=O)CCC1)=O

-20°C

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Peptide