UFP-101 - CAS 849024-68-6

Potent, selective and competitive silent antagonist for the NOP opioid receptor. Binds to NOP with high affinity (pKi = 10.24) and displays > 3000-fold selectivity over δ, μ and κ opioid receptors. Antinociceptive and opposes the action of nociceptin in vivo.

Opioid Receptor

Neuroscience, Endocrinology/Hormones, GPCR/G Protein

849024-68-6

C82H138N32O21

1908.19

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-20°C

Ice Packs

Peptide