UniPR500 - CAS 2085767-98-0

UniPR500, a derivative of UniPR129, is a competitive antagonist for the EphA2 receptor, with a Ki of 0.78 μM. It reduces the binding of biotinylated Ephrin-A1 to EphA2 in a dose-dependent manner, exhibiting an IC50 value of 1.1 μM.

Ephrin Receptor

Tyrosine Kinase/Adaptors

2085669

C36H51N3O4

589.808

C[C@@]12[C@]([C@]3([C@@]([C@]4(C)[C@](CC3)(CC(=NO)CC4)[H])(CC1)[H])[H])(CC[C@@]2([C@@H](CCC(N[C@@H](CC=5C=6C(NC5)=CC=CC6)CC(O)=O)=O)C)[H])[H]

-20°C

Ice Packs

Small Compound