VA5 TG2 inhibitor - CAS 2088001-24-3

VA5 is an transamidase inhibitor by direct binding at the transamidase site. VA5 also inhibits GTP-binding activities. It interaction at the transamidase site locks the protein in the extended/open conformation to disorganize/inactivate the GTP binding/GTPase site.

Others, BTK

Others, Angiogenesis, Tyrosine Kinase/Adaptors

2087974

C31H34N4O8

590.62

Oc1ccc2cc(C(=O)N3CCN(CC3)C(=O)[C@H](CCCCNC(=O)C=C)NC(=O)OCc3ccccc3)c(=O)oc2c1

-20°C

Ice Packs

Small Compound