VGSC blocker-1 - CAS 2230472-55-4

VGSC blocker-1 is a powerful small molecule that serves as a blocker for the neonatal isoform of the VGSC subtype known as Nav1.5 (nNav1.5) . It effectively blocks INa peak currents by 34.9% at a concentration of 1 μM, and demonstrates a 0.3% inhibition of cell invasion at the same concentration in the MDA-MB-231 human breast cancer cell line, without compromising cell viability.

Others, Sodium Channel

Others, Membrane transporter/Ion channel

2230472-55-4

C24H32F2N2

386.52

Fc1ccc(cc1)C(CCCNCCCN1CCCCC1)c1ccc(F)cc1

-20°C

Ice Packs

Small Compound