YM022 - CAS 145084-28-2

YM022 is a highly effective and selective gastrin/cholecystokinin (CCK) -B receptor antagonist. YM022 can inhibit gastrin-induced gastric acid secretion and histidine decarboxylase activation in vivo. YM022 shows the Ki values of 68 pM and 63 nM for CCK-B and CCK-A receptor, respectively.

CCR

GPCR/G Protein, Immunology/Inflammation, Microbiology/Virology

145054

C32H28N4O3

516.59

Cc1cccc(NC(=O)N[C@@H]2N=C(c3ccccc3)c3ccccc3N(CC(=O)c3ccccc3C)C2=O)c1

-20°C

Ice Packs

Small Compound